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60

抑制剂 & 化合物

20

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Cat. No. Product Name Target Signaling Pathways
T38240 2,6-Dichlorodiphenylamine

Antibacterial Microbiology/Virology
2,6-Dichlorodiphenylamine 是双氯芬酸钠的一种结构类似物,显示出抗白色念珠菌活性。2,6-Dichlorodiphenylamine 是非选择性抗炎剂,为COX 的抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50分别为 4 和 1.3 nM。
T27617 Inz-1

P450 Metabolism
Inz-1 是一种有效的真菌特异性线粒体细胞色素 bc1 抑制剂,对酵母和人类的 IC50 分别为 8.092 和 45.320 μM。 Inz-1 可逆转氟康唑或其他三唑类抗真菌药对致病性真菌白色念珠菌的耐药性。
T21678 3MB-PP1

PLK Cell Cycle/Checkpoint
3MB-PP1是嘌呤类似物,是一种 Polo 样激酶 1 (Plk1) 抑制剂。在表达类似物敏感的 Plk1 等位基因的细胞中,3MB-PP1 通过靶向 Plk1 阻断有丝分裂进程和细胞分裂。3MB-PP1 特异性抑制类似物敏感的 Ssn3 (Cdk8)。3MB-PP1 抑制 Leu93 突变 Zipper-interacting protein kinase(Leu93-ZIPK),IC50为2 μM。3MB-PP1 可用于细胞分裂和白色念珠菌 (Candida albicans) 菌丝形成的研究。
T19717 Cyclo-L-Trp-L-Trp

Antifungal Microbiology/Virology
Cyclo-L-Trp-L-Trp 是一种广谱抗真菌剂。它还诱导组蛋白的高度乙酰化。
T17022 Tebuconazole

P450; Antifungal Metabolism; Microbiology/Virology
Tebuconazole 是一种农用唑类杀菌剂,可抑制 CYP51,对白色念珠菌 CYP51 和truncated Homo sapiens CYP51 的IC50分别为 0.9 和 1.3 μM。
T9602 Monocaprin

Anti-infection; Antibacterial Microbiology/Virology
Monocaprin 是癸酸的 1-单甘油酯,对包膜病毒、某些细菌和酵母白色念珠菌具有抗菌活性。
T16412 Oteseconazole

VT-1161

P450; Antifungal Metabolism; Microbiology/Virology
Oteseconazole (VT-1161) 是一种口服有效的抗真菌剂,结合并抑制白色念球菌的 CYP51,Kd 值小于 39 nM。
T8536 Filastatin

Antifungal Microbiology/Virology
Filastatin 是一种长效的白色念珠菌丝状体抑制剂,具有强大的抗真菌作用。它抑制真菌与聚苯乙烯和人类细胞的粘附,从酵母到菌丝的形态转变,抑制菌丝特异性 HWP1 启动子。
T77686 1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone

Antifungal Microbiology/Virology
1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone 具有广谱的抗真菌活性,对白色念珠菌、黑曲霉、铜绿假单胞菌、金黄色葡萄球菌等具有抑制作用。
T61502 Antifungal agent 32

Antifungal agent 32 (compound 1a) is a highly effective antifungal compound. It displays strong inhibitory activity against Candida albicans filamentation and biofilm formation, as well as inhibiting the morphological switching of Candida albicans and its adherence to epithelial cells. This makes Antifungal agent 32 a valuable tool for research on Candida albicans infections [1].
T13787 N-563

Others Others
N-563 promotes resistance to Candida albicans infection in mice
T35297 ZD 0870

D 0870,D0870,ZD0870

ZD 0870, used to treat infections caused by fluconazole-resistant candida albicans.
T28596 RO-09-4609

RO 09-4609,RO09-4609,RO 094609,RO-094609

RO-09-4609 is a potent and selective inhibitor of Candida albicans N-myristoyltransferase (CaNmt).
T81494 PhD3

PhD3是源自猴血白细胞的抗菌肽,具备针对细菌和(Candida albicans)的抗菌活性。
T81495 PhD2

PhD2是一种源自猴血白细胞的抗菌肽,对细菌与(真菌)Candida albicans显示出抗生活性。
T81496 PhD1

PhD1是一种抗菌肽,源自猴血白细胞,对细菌和白色念珠菌(Candida albicans)具有抗菌活性。
T81493 PhD4

PhD4,源自猴血白细胞的抗菌肽,对细菌和真菌(Candida albicans)均显示活性。
T25342 Discobahamin A

Discobahamin A is a bioactive peptide isolated from a new species of the Bahamian deep water marine sponge Discodermia. It is a growth of Candida albicans inhibitor.
T25343 Discobahamin B

Discobahamin B is a bioactive peptide isolated from a new species of the Bahamian deep water marine sponge Discodermia. It is a growth of Candida albicans inhibitor.
T80629 2-Dodecanol

2-Dodecanol有效抑制了C. albicans的菌丝形成和SIR2基因的表达。
T64235 Antifungal agent 25

Antifungal agent 25 是一种有效的、广谱的、体内具有代谢稳定性的抗真菌剂。Antifungal agent 25 对白色念珠菌和耐氟康唑的白色念珠菌都表现出抗真菌效果。
T62098 Antifungal agent 28

Antifungal agent 28 (化合物 18) 是一种选择性的、有效的抗真菌剂。Antifungal agent 28 可以破坏成熟念珠菌生物膜,能够抑制白念珠菌和非白念珠菌的致病性菌株,包括耐氟康唑菌株。Antifungal agent 28 对隐球菌和曲霉菌株也具有抑制作用。
T63755 Antitubercular agent-22

Antitubercular agent-22 (Compound 2) 是有效的抗念珠菌和抗结核剂,能够作用于 Candida albicansMTCC 3017 (MIC: 2.34 μg/ml) 和 M. tuberculosis(H37Rv) (MIC: 2 μg/ml)。
T69051 Aculeacin A

Aculeacin A is used to study mutations that lead to antibiotic resistance in Saccharomyces cerevisiae, the inhibition of Candida albicans and the morphogenetic transformation of Candida albicans when treated. Aculeacin A is a lipopeptide that inhibits β-glucan synthesis in yeasts. The inhibition is due to the selective blockage of glucan synthase. Aculeacin A, an amphophilic antibiotic, inhibits the biosynthesis of β−glucan by selective blockage of β(1→3) glucan synthase.
T76470 GVLSNVIGYLKKLGTGALNAVLKQ

GVLSNVIGYLKKLGTGALNAVLKQ 是一种具有 24 个氨基酸的抗菌肽。 GVLSNVIGYLKKLGTGALNAVLKQ 可能形成 α 螺旋。GVLSNVIGYLKKLGTGALNAVLKQ (PGQ) 对革兰氏阴性菌、革兰氏阳性菌和酵母Candida albicans 具有抗性。
T63525 Antitubercular agent-23

Antitubercular agent-23 是有效的抗念珠菌及抗结核剂,能够作用于 Candida albicansMTCC 3017 (MIC: 1.1 μg/ml) 和 M. tuberculosis(H37Rv) (MIC: 1 μg/ml)。
T10311 Amphotericin X1

两性霉素 X1

Others Others
Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, C.parapsilosis 937A, Aspergillus niger 57A and A.fumigatus (MICs: 1 μg/mL, 1 μg/mL, 8 μg/mL, 2
T80932 Tritrpticin

Tritrpticin是一种来源于猪骨髓的抗菌肽,对Aspergillus fumigatus和Candida albicans表现出抗菌活性,其最小抑菌浓度(MIC)分别为250和1000 μg/ml。
T62159 Antifungal agent 24

Antifungal agent 24 (Compound 6) 是一种抗真菌剂,能够抑制白色念珠菌 (MIC: 0.03 μg/ml)。
T63064 Antibacterial agent 100

Antibacterial agent 100 (Compound 7c) 是一种抗细菌和真菌剂,能够作用于 Staphylococcus aureus (MIC: 4 μg/mL)、Candida albicans (MIC: 4 μg/mL) 和 Cryptococcus neoformans (MIC: 8 μg/mL)。
T82834 Bombinin-BO1

Bombinin-BO1是一种蟾蜍皮肤分泌物中的抗菌肽,它对大肠杆菌(Escherichia coli)、金黄色葡萄球菌(Staphylococcus aureus)和白色念珠菌(Candida albicans)显示出抗生活性,其最小抑菌浓度(MIC)值分别为64 mg/L, 64 mg/L和128 mg/L。
T80296 SP-B peptide

SP-B peptide 是具有抗真菌活性的抗菌肽,有效针对新型隐球菌、白色念珠菌及烟曲霉菌株。
T61398 Chitin synthase inhibitor 3

Chitin synthase inhibitor 3 (compound 2d) 是一种高效的chitin synthase抑制剂,具有0.16 mM的IC50值,并对candida albicans显示出1 μg/mL的MIC,表现出抗真菌活性。
T75176 Antifungal agent 53

Antifungal agent 53 (A03) 是一种有效的白色念珠菌 CYP51抑制剂,具有抗真菌活性。Antifungal agent 53 阻止真菌生物膜的形成。Antifungal agent 53 也显示出良好的安全性。
T82835 Bombinin H-BO1

Bombinin H-BO1 是源自蟾蜍皮肤分泌物的抗菌肽,对白色念珠菌有效,其MIC值达256 mg/L。
T39322 Temporin A

Temporin A, a short alpha-helical antimicrobial peptide derived from the skin of Rana temporaria, exhibits a wide-ranging efficacy against Gram-positive bacteria. It directly interacts with the cell membrane of microorganisms and remains non-toxic to erythrocytes at antimicrobial concentrations. Additionally, Temporin A demonstrates antifungal properties against yeast-like Candida albicans.
T74273 Antifungal agent 52

Antifungal agent 52 (compound 6c) 是四唑衍生物。Antifungal agent 52 抑制麦角固醇 的合成。Antifungal agent 52 对白色念珠菌表现出显着的抗真菌活性 Antifungal agent 52 影响白色念珠菌基底细胞膜通透性。
T74831 Antifungal agent 51

Antifungal agent 51 (5c) 具有强效的抗真菌活性,尤其是对白色念珠菌 FDC 151 、近平滑念珠菌 ATCC 22019 和热带假丝酵母 FDC 138,MIC 值小于 0.063 μg/mL,而对细胞的毒性较低,无致癌性。
T64127 VT-1598

VT-1598 是一种新型的、选择性的、口服居于活力的 fungal CYP51 抑制剂。VT-1598 对白色念珠菌表现出抗真菌效果。
T75178 Antifungal agent 55

Antifungal agent 55 (compound A07) 是一种抗氟康唑 耐药菌株的强效抗真菌剂。Antifungal agent 55 比咪康唑 更有效。Antifungal agent 55 抑制白色念珠菌的 MIC 值为 0.25-1 μg/mL。
T74959 Antifungal agent 41

Antifungal agent 41 (compound B01) 是一种抗真菌剂。Antifungal agent 41 在体内外表现出对白假丝酵母菌的抗性。Antifungal agent 41 可以用于侵袭性真菌感染的研究。
T75181 Antifungal agent 58

Antifungal agent 58 (compound A21) 是一种抗氟康唑 耐药菌株的强效抗真菌剂。Antifungal agent 58 比咪康唑 更有效。Antifungal agent 58 抑制白色念珠菌的 MIC 值为 0.06-8 μg/mL。
T75179 Antifungal agent 56

Antifungal agent 56 (compound A09) 是一种抗氟康唑 耐药菌株的强效抗真菌剂。Antifungal agent 56 比咪康唑 更有效。Antifungal agent 56 抑制白色念珠菌的 MIC 值为 0.03-0.25 μg/mL。
T75180 Antifungal agent 57

Antifungal agent 57 (compound A19) 是一种抗氟康唑 耐药菌株的强效抗真菌剂。Antifungal agent 57 比咪康唑 更有效。Antifungal agent 57 抑制白色念珠菌的 MIC 值为 0.5-2 μg/mL。
T62211 Antifungal agent 33

Antifungal agent 33 (compound 4e) 是一种有效的抗真菌剂。Antifungal agent 33 对白念珠菌具有明显的抗真菌作用 (MIC: 16 μg/ml)。Antifungal agent 33 能够较强的抑制羊毛甾醇 14α-去甲基化酶 (CYP51) (IC50: 0.19 μg/ml)。
T79551 Antifungal agent 69

Antifungalagent 69 (compound 13),作为一种丁子香酚-咪唑类化合物,对白色念珠菌表现出有效的抗真菌活性,其MIC值为4.6 μM,并未展现显著的细胞毒性。此外,该化合物能够干预真菌的麦角甾醇生物合成路径。
T75177 Antifungal agent 54

Antifungal agent 54 (compound A05) 是一种抗氟康唑 耐药菌株的强效抗真菌剂。Antifungal agent 54 比咪康唑 更有效。Antifungal agent 54 抑制白色念珠菌的 MIC 值为 0.25-1 μg/mL。
T83069 Antifungal agent 75

Antifungalagent 75 (compound 6r) 是针对白色念珠菌有效的抗真菌剂。该化合物通过显著抑制生物膜形成、增加细胞膜通透性、降低麦角甾醇水平并破坏膜结构,从而破坏细胞结构完整性,发挥其抗真菌活性。
T79467 Antifungal agent 60

Antifungalagent 60(compound 16)是一种抑制麦角甾醇生物合成的广谱抗真菌剂。它能够有效抑制包括7种人类致病真菌、2种耐氟康唑的白色念珠菌分离株以及2种多重耐药的耳念珠菌分离株。
T60684 FBA-IN-1

FBA-IN-1 (compound 2a11) 是首创的,对白色念珠菌的 1,6-二磷酸果糖醛缩酶 (CaFBA) 的共价变构抑制剂。此外,FBA-IN-1 以 MIC80为 1 μg/mL,抑制唑类耐药菌株 103 的生长。

化合物

2,6-Dichlorodiphenylamine
Cat.No: T38240
Synonym:
Target: Antibacterial
Inz-1
Cat.No: T27617
Synonym:
Target: P450
3MB-PP1
Cat.No: T21678
Synonym:
Target: PLK
Cyclo-L-Trp-L-Trp
Cat.No: T19717
Synonym:
Target: Antifungal
Tebuconazole
Cat.No: T17022
Synonym:
Target: P450, Antifungal
Monocaprin
Cat.No: T9602
Synonym:
Target: Anti-infection, Antibacterial
Oteseconazole
Cat.No: T16412
Synonym: VT-1161
Target: P450, Antifungal
Filastatin
Cat.No: T8536
Synonym:
Target: Antifungal
1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone
Cat.No: T77686
Synonym:
Target: Antifungal
Antifungal agent 32
Cat.No: T61502
Synonym:
Target:
N-563
Cat.No: T13787
Synonym:
Target: Others
ZD 0870
Cat.No: T35297
Synonym: D 0870,D0870,ZD0870
Target:
RO-09-4609
Cat.No: T28596
Synonym: RO 09-4609,RO09-4609,RO 094609,RO-094609
Target:
PhD3
Cat.No: T81494
Synonym:
Target:
PhD2
Cat.No: T81495
Synonym:
Target:
PhD1
Cat.No: T81496
Synonym:
Target:
PhD4
Cat.No: T81493
Synonym:
Target:
Discobahamin A
Cat.No: T25342
Synonym:
Target:
Discobahamin B
Cat.No: T25343
Synonym:
Target:
2-Dodecanol
Cat.No: T80629
Synonym:
Target:
Antifungal agent 25
Cat.No: T64235
Synonym:
Target:
Antifungal agent 28
Cat.No: T62098
Synonym:
Target:
Antitubercular agent-22
Cat.No: T63755
Synonym:
Target:
Aculeacin A
Cat.No: T69051
Synonym:
Target:
GVLSNVIGYLKKLGTGALNAVLKQ
Cat.No: T76470
Synonym:
Target:
Antitubercular agent-23
Cat.No: T63525
Synonym:
Target:
Amphotericin X1
Cat.No: T10311
Synonym: 两性霉素 X1
Target: Others
Tritrpticin
Cat.No: T80932
Synonym:
Target:
Antifungal agent 24
Cat.No: T62159
Synonym:
Target:
Antibacterial agent 100
Cat.No: T63064
Synonym:
Target:
Bombinin-BO1
Cat.No: T82834
Synonym:
Target:
SP-B peptide
Cat.No: T80296
Synonym:
Target:
Chitin synthase inhibitor 3
Cat.No: T61398
Synonym:
Target:
Antifungal agent 53
Cat.No: T75176
Synonym:
Target:
Bombinin H-BO1
Cat.No: T82835
Synonym:
Target:
Temporin A
Cat.No: T39322
Synonym:
Target:
Antifungal agent 52
Cat.No: T74273
Synonym:
Target:
Antifungal agent 51
Cat.No: T74831
Synonym:
Target:
VT-1598
Cat.No: T64127
Synonym:
Target:
Antifungal agent 55
Cat.No: T75178
Synonym:
Target:
Antifungal agent 41
Cat.No: T74959
Synonym:
Target:
Antifungal agent 58
Cat.No: T75181
Synonym:
Target:
Antifungal agent 56
Cat.No: T75179
Synonym:
Target:
Antifungal agent 57
Cat.No: T75180
Synonym:
Target:
Antifungal agent 33
Cat.No: T62211
Synonym:
Target:
Antifungal agent 69
Cat.No: T79551
Synonym:
Target:
Antifungal agent 54
Cat.No: T75177
Synonym:
Target:
Antifungal agent 75
Cat.No: T83069
Synonym:
Target:
Antifungal agent 60
Cat.No: T79467
Synonym:
Target:
FBA-IN-1
Cat.No: T60684
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1388 Fluconazole

氟康唑,UK-49858

Antibiotic; Antifection; Antifungal Microbiology/Virology
Fluconazole (UK-49858) 是一种对多种真菌具有活性的三唑类抗真菌剂,抑制 C. albicansCandida kefyr 的 IC99为 0.20 μg/mL 至 0.39 μg/mL。
T14046 Anandamide

花生四烯酸乙醇胺,(5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide

Cannabinoid Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism
Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide) 是一种免疫调节剂,通过大麻素受体 CB1 和 CB2 起作用,还通过中枢神经系统中的其他靶点起作用,如 GPR18/GPR55。
T7029 Pseudolaric Acid C

Antifungal Microbiology/Virology
Pseudolaric Acid C 是一种从Pseudolarix kaempferiGorden 根皮部中分离的二萜酸,对白色念珠菌有较弱的抗真菌活性。
TN1651 Furanodiene

Apoptosis; PARP; Reactive Oxygen Species; Caspase; CDK; P-gp Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Proteases/Proteasome
Furanodiene 是从姜黄中提取的一种萜类天然产物,可抑制外排转运蛋白Pgp 功能并降低 Pgp 蛋白水平。它通过抗血管生成和诱导ROS 产生,DNA 链断裂和细胞凋亡发挥抗癌作用。
T1678 Nystatin

Stamycin,Fungicidin,制霉菌素,Nystavescent

Apoptosis; Antibiotic; Antifungal Apoptosis; Microbiology/Virology
Nystatin (Fungicidin) 是一种口服对酵母和支原体有效的多烯类抗真菌抗生素。它能增加质膜对包括氯离子等小单价离子的通透性。它可部分阻止 Oxaliplatin 诱导的脂筏聚集、DR4 和 DR5 聚集的胆固醇隔离试剂,减少细胞凋亡。
T0011 2-Phenylethanol

苯乙醇,Phenethyl alcohol,2-Phenylethyl alcohol,Benzyl carbinol,Phenylethanol,Benzeneethanol

Others; Virus Protease; Antibacterial; Antibiotic Microbiology/Virology; Others
2-Phenylethanol (Phenylethanol) 是从玫瑰、风笛、阿勒颇松、桔子花等多种物种中提取得到的一种无色液体。它有一种使人感到愉悦的气味,也是一种从真菌Candida albicans 产生的自体抗生素。它可用作香皂中的防腐剂,也用作香烟添加剂。
T25718 Lichesterol

Lichesterol is extracted from polyene antibiotic-resistant Candida albicans.
TN2032 Pachypodol

霍香黃酮醇

Antifection Microbiology/Virology
Pachypodol has antibacterial and antifungal activities against Bacillus subtilis, Staphylococcus aureus, Staphylococcus faecalis, Echerichia coli, Pseudomonas aeruginosa, Candida albicans, Candida krusei and Candida galabrata.
TN1561 Dehydroglaucine

Antifection Microbiology/Virology
Dehydroglaucine is an acetylcholinesterase inhibitor, it shows antimicrobial activity against Staphylococcus aureus, Mycobacterium smegmatis, Candida albicans, and Aspergillus niger.
TN2492 1,4,5,6-Tetrahydroxy-7,8-diprenylxanthone

Others Others
1,4,5,6-Tetrahydroxy-7,8-diprenylxanthone has moderate cytotoxicities against breast cancer (MDA-MB-435S) and lung adenocarcinoma (A549) cell lines, but lacks antifungal activity against Candida albicans.
TN3400 Altechromone A

Antifection Microbiology/Virology
Altechromone A has antimicrobial activity, it is active against Bacillus subtilis, Escherichia coli, Pseudomonas fluorescens and Candida albicans with the MICs of 3.9, 3.9, 1.8, and 3.9 ug/ml, respectively.
T28379 PF-1163B

PF1163B,(-)-PF1163B,PF 1163B

PF-1163B is an antifungal agent form Penicillium sp. II. PF-1163B inhibits ergosterol (ERG) synthesis with IC50 value of 34 ng/ml. PF-1163B showed potent growth inhibitory activity against pathogenic fungal strain Candida albicans but did not show cytotox
T80335 Maximin H3

Maximin H3,源自中华红腹蟾蜍Bombina maxima皮肤分泌,为一种抗菌肽。对Escherichia coli ATCC 25922、Staphylococcus aureus ATCC 2592、Bacillus pyocyaneus CMCC B1010 及Candida albicans ATCC 2002表现出显著抗性,其MIC值依次为20, 10, 20, 5 μg/ml。
T79931 Mutanocyclin

Mutanocyclin 作为一种效能显著的抗真菌剂,能够抑制白色念珠菌 (C. albicans) 的丝状形成,并下调 HWP1、ECE1、FLO8、TEC1 基因的 mRNA 表达水平。此外,Mutanocyclin 在体外小鼠模型中亦能有效抑制酵母形态的发展。
T80349 Maximin H4

Maximin H4是一种来自中华红腹蟾蜍(Bombina maxima)皮肤分泌物的抗菌肽,具有针对Escherichia coli ATCC25922、Staphylococcus aureus ATCC2592、Bacillus pyocyaneus CMCCB1010和Candida albicans ATCC2002的抗菌活性。其最小抑菌浓度(MIC)值依次为12、6、12、6 μg/ml。
T80334 Maximin H2

Maximin H2,源自中华红腹蟾蜍(Bombina maxima)皮肤分泌物的抗菌肽,对Escherichia coli ATCC25922、Staphylococcus aureus ATCC2592、Bacillus pyocyaneus CMCCB1010及Candida albicans ATCC2002展示了明显的抗菌活性。其最小抑菌浓度(MIC)值依序为20、2、4、2 μg/ml。
T69225 Verrucarin J

Muconomycin B

Verrucarin J (Muconomycin B) 是Myrothecium 真菌家族的代谢物。Verrucarin J 诱导活性氧 (ROS) 生成和癌细胞系凋亡 (apoptosis),例如 A549、HCT 116 和 SW-620 细胞。Verrucarin J 具有抗Candida albicans 和Mucor miehei 的活性。Verrucarin J 抑制沙粒病毒 Junin (JUNV) 产量,IC50为 1.2 ng/mL。
T80332 Maximin H1

Maximin H1是一种抗菌肽,由中华红腹蟾蜍(Bombina maxima)皮肤分泌物提取得到。该化合物对Escherichia coli ATCC 25922、Staphylococcus aureus ATCC 25923、Bacillus pyocyaneus CMCC B1010和Candida albicans ATCC 2002表现出抗菌活性,其最小抑菌浓度(MIC)值分别为9、4.5、9、4.5 μg/ml。
T79008 Ys-II

Ys-II (Compound 1)为源于丝兰(Yucca elephantipe)茎部的螺甾烷醇糖苷,具备针对白色念珠菌和新型隐球菌(Cryptococcus neoformans)的抗真菌效力(IC50分别为5和6μg/mL)。
TN4471 Lysicamine

IL Receptor; Antifection Immunology/Inflammation; Microbiology/Virology
Lysicamine shows significant antioxidant capacity in the ORAC(FL) assay and it is active against S. epidermidis and C. dubliniensis, with MIC values in the range 12.5-100 microg mL(-1). Lysicamine has antimicrobial and anti-inflammation activity, the mini

天然产物

Fluconazole
Cat.No: T1388
Synonym: 氟康唑,UK-49858
Target: Antibiotic, Antifection, Antifungal
Anandamide
Cat.No: T14046
Synonym: 花生四烯酸乙醇胺,(5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide
Target: Cannabinoid Receptor, Endogenous Metabolite
Pseudolaric Acid C
Cat.No: T7029
Synonym:
Target: Antifungal
Furanodiene
Cat.No: TN1651
Synonym:
Target: Apoptosis, PARP, Reactive Oxygen Species, Caspase, CDK, P-gp
Nystatin
Cat.No: T1678
Synonym: Stamycin,Fungicidin,制霉菌素,Nystavescent
Target: Apoptosis, Antibiotic, Antifungal
2-Phenylethanol
Cat.No: T0011
Synonym: 苯乙醇,Phenethyl alcohol,2-Phenylethyl alcohol,Benzyl carbinol,Phenylethanol,Benzeneethanol
Target: Others, Virus Protease, Antibacterial, Antibiotic
Lichesterol
Cat.No: T25718
Synonym:
Target:
Pachypodol
Cat.No: TN2032
Synonym: 霍香黃酮醇
Target: Antifection
Dehydroglaucine
Cat.No: TN1561
Synonym:
Target: Antifection
1,4,5,6-Tetrahydroxy-7,8-diprenylxanthone
Cat.No: TN2492
Synonym:
Target: Others
Altechromone A
Cat.No: TN3400
Synonym:
Target: Antifection
PF-1163B
Cat.No: T28379
Synonym: PF1163B,(-)-PF1163B,PF 1163B
Target:
Maximin H3
Cat.No: T80335
Synonym:
Target:
Mutanocyclin
Cat.No: T79931
Synonym:
Target:
Maximin H4
Cat.No: T80349
Synonym:
Target:
Maximin H2
Cat.No: T80334
Synonym:
Target:
Verrucarin J
Cat.No: T69225
Synonym: Muconomycin B
Target:
Maximin H1
Cat.No: T80332
Synonym:
Target:
Ys-II
Cat.No: T79008
Synonym:
Target:
Lysicamine
Cat.No: TN4471
Synonym:
Target: IL Receptor, Antifection
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